SCHEMBL5766014

SCHEMBL5766014

NCCCOc1ccc2nccc(NC(=O)OC3CCN(CCc4nc5c(F)cccc5[nH]4)CC3)c2n1

nearest known ligand 0.41

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 13/20 0.41
SLC40A1 Q9NP59 4/20 0.39
KCNH2 Q12809 3/20 0.38
CHRM2 P08172 2/20 0.38
CHRM1 P11229 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14573161 0.91 SLC40A1 (0.40) SLC40A1KCNH2
SCHEMBL5765657 0.91 KCNH2 (0.47) SLC40A1KCNH2
SCHEMBL14573148 0.81 KCNH2 (0.47) SLC40A1KCNH2
SCHEMBL5657252 0.81 SLC40A1 (0.37) SLC40A1KCNH2
SCHEMBL5774180 0.80 KCNH2 (0.42) SLC40A1KCNH2
SCHEMBL6661601 0.74 KCNH2 (0.45) SLC40A1KCNH2
SCHEMBL5764918 0.70 KCNH2 (0.45) CHRM3KCNH2
SCHEMBL5657093 0.69 CHRNA7 (0.47) SLC40A1
SCHEMBL5765881 0.69 KCNH2 (0.45) KCNH2
SCHEMBL5764847 0.68 KCNH2 (0.48) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1392686-B1 BICYCLIC NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVES FOR USE AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2006-10-18 EP claimed