SCHEMBL1458449

SCHEMBL1458449

O=C(O)c1cccc(-c2ccc(C3CN(S(=O)(=O)c4ccccc4I)C(=O)N3c3ccccc3)cc2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.39
CMA1 P23946 2/20 0.37
CTSG P08311 1/20 0.37
ACLY P53396 1/20 0.35
TDP2 O95551 1/20 0.34
MCL1 Q07820 1/20 0.34
PDE5A O76074 1/20 0.34
AKR1C3 P42330 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
PFKFB3 Q16875 1/20 0.33
GRIA2 P42262 1/20 0.33
KCNH2 Q12809 1/20 0.33
NPC1 O15118 1/20 0.33
MITF O75030 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
NFKB1 P19838 1/20 0.33
APOBEC3A P31941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1459376 0.93 CMA1 (0.38) KMOCMA1CTSGAKR1C3PFKFB3
SCHEMBL1348640 0.88 CMA1 (0.44) KMOCMA1CTSGACLYMCL1
SCHEMBL1458988 0.81 F10 (0.31) MCL1KMT2A
SCHEMBL1348740 0.81 CMA1 (0.45) KMOCMA1CTSGMCL1AKR1C3
SCHEMBL1347258 0.79 CTSG (0.46) CMA1CTSGMCL1ALDH1A1RAB9A
SCHEMBL1348608 0.79 MCL1 (0.43) CMA1CTSGMCL1AKR1C3ALDH1A1
SCHEMBL15841996 0.74 BCL9 (0.37) CMA1CTSGMCL1AKR1C3
SCHEMBL1348917 0.74 GRIA2 (0.43) GRIA2ALDH1A1RAB9AKMT2ASMN1; SMN2
SCHEMBL27807888 0.72 ACMSD (0.40) CMA1CTSGACLYMCL1AKR1C3
SCHEMBL15841773 0.70 BCL9 (0.37) MCL1AKR1C3LMNAGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2288594-A1 IMIDAZOLIDINE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2011-03-02 EP disclosed
WO-2009150109-A1 IMIDAZOLIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2009-12-17 WO disclosed