SCHEMBL14595331

SCHEMBL14595331

CCCc1ccc(Cl)c(NCc2ccc(-c3nccc(NCC4CC4)n3)cc2)c1CCC

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 16/20 0.44
DYRK1A Q13627 8/20 0.41
CLK1 P49759 2/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CLK2 P49760 1/20 0.38
DYRK1B Q9Y463 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12160418 0.76 CLK4 (0.41) CLK4DYRK1ACLK1KDM4EALDH1A1
SCHEMBL2586735 0.71 ADRB2 (0.47) CLK4DYRK1ACLK1KDM4EALDH1A1
Succinic Acid SCHEMBL2587865 0.71 ALDH1A1 (0.38) CLK4DYRK1ACLK1KDM4EALDH1A1
SCHEMBL13685572 0.69 CLK4 (0.34) CLK4DYRK1ACLK1KDM4EALDH1A1
SCHEMBL2579999 0.67 ACACB (0.48) CLK4CLK1ALDH1A1CYP1A2CYP3A4
SCHEMBL11948255 0.66 MAOA (0.31)
SCHEMBL14488434 0.64 CLK4 (0.49) CLK4DYRK1ACLK1ALDH1A1CYP1A2
SCHEMBL2588748 0.63 GNRHR (0.46)
SCHEMBL11948250 0.62
SCHEMBL13825303 0.62

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed