SCHEMBL14596409

SCHEMBL14596409

C=C(Br)c1ccc(Br)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
CYP2A6 P11509 1/20 0.47
CA1 P00915 3/20 0.46
CA2 P00918 3/20 0.46
ALOX15 P16050 2/20 0.43
GSK3B P49841 2/20 0.42
OGG1 O15527 1/20 0.41
LMNA P02545 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5049280 0.79 MAPT (0.55) CES2CES1CYP2A6CA1CA2
SCHEMBL21679933 0.79 CES2 (0.52) CES2CES1CYP2A6CA1CA2
SCHEMBL6343638 0.79 MAPT (0.55) CES2CES1CYP2A6CA1CA2
SCHEMBL17547225 0.77 CES2 (0.50) CES2CES1CYP2A6CA1CA2
SCHEMBL8587179 0.74 CES2 (0.48) CES2CES1CA1CA2RAB9A
SCHEMBL942286 0.74 CES2 (0.48) CES2CES1CYP2A6CA1CA2
SCHEMBL206782 0.74 CES2 (0.48) CES2CES1CYP2A6CA1CA2
SCHEMBL6036757 0.74 CES2 (0.48) CES2CES1CYP2A6CA1CA2
SCHEMBL7922645 0.74 CES2 (0.48) CES2CES1CYP2A6CA1CA2
SCHEMBL12449040 0.74 MAPT (0.32) CES2CES1GSK3BLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113511972-A (E) Preparation method of (E) -4-aryl-2, 2-difluoro-3-butenoic acid derivative 昆明理工大学 2021-10-19 CN disclosed
WO-2007024922-A1 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS IRM LLC (BM) 2007-03-01 WO disclosed