SCHEMBL14599876

SCHEMBL14599876

C=CC[C@H](O)C#Cc1csc(C)n1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 19/20 0.46
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5567017 1.00 GRM5 (0.46) GRM5CYP1A2CYP2D6
SCHEMBL5567321 0.71 GRM5 (0.46) GRM5CYP1A2CYP2D6
SCHEMBL15494395 0.71 GRM5 (0.53) GRM5CYP1A2CYP2D6
SCHEMBL3353813 0.67 GRM5 (0.68) GRM5CYP1A2CYP2D6
SCHEMBL729985 0.67 KMT2A (0.38) GRM5
SCHEMBL14006347 0.66
SCHEMBL12230330 0.65 GRM5 (0.32) GRM5
SCHEMBL8024334 0.65 GRM5 (0.32) GRM5
SCHEMBL8024330 0.65 GRM5 (0.32) GRM5
SCHEMBL14587140 0.65 GRM5 (0.32) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7157595-B2 Degradation of epothilones HELMHOLTZ-ZENTRUM FUR INFEKTIONSFORSCHUNG GMBH (DE) 2007-01-02 US disclosed