SCHEMBL14600779

SCHEMBL14600779

Cc1cccc(-c2cnoc2-c2c[nH]c(C(=O)NC[C@@H]3CCCO3)n2)c1F

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
RAB9A P51151 2/20 0.46
NPC1 O15118 2/20 0.46
HPGD P15428 4/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
GAA P10253 2/20 0.45
CYP2C9 P11712 1/20 0.45
ALDH1A1 P00352 6/20 0.45
GSK3B P49841 1/20 0.44
KCNH2 Q12809 1/20 0.44
TSHR P16473 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 1/20 0.43
TP53 P04637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.42
ATM Q13315 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600777 0.92 GSK3B (0.53) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14600753 0.87 GSK3B (0.53) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14278769 0.77 GSK3B (0.55) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14286127 0.74 GSK3B (0.56) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14600773 0.73 RAB9A (0.47) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL10067976 0.73 GSK3B (0.44) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL10067975 0.73 ALDH1A1 (0.46) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14600763 0.73 GSK3B (0.44) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL14600774 0.73 GSK3B (0.45) MEN1KMT2ARAB9ANPC1HPGD
SCHEMBL10067977 0.73 GSK3B (0.47) MEN1KMT2ARAB9ANPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7169800-B2 Imidazole compositions useful as inhibitors of protein kinases VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-01-30 US disclosed