SCHEMBL14601259

SCHEMBL14601259

CC(=O)c1ccc(C2CCN(C(=O)c3cccc(Oc4ccc(C)cc4)c3)CC2)cc1

nearest known ligand 0.67

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 11/20 0.67
PARP14 Q460N5 7/20 0.67
MAPT P10636 2/20 0.59
CRHBP P24387 1/20 0.59
HTT P42858 1/20 0.59
CRHR2 Q13324 1/20 0.59
MGLL Q99685 5/20 0.53
NPC1 O15118 1/20 0.52
HSD11B1 P28845 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL903593 0.83 MAPT (0.85) PARP10PARP14MAPTCRHBPHTT
SCHEMBL257897 0.80 MEN1 (0.64) PARP10PARP14MAPTCRHBPHTT
SCHEMBL24489414 0.76 MAPT (0.66) PARP10PARP14MAPTCRHBPHTT
SCHEMBL25910311 0.76 MAOB (0.63) PARP10PARP14MAPTCRHBPHTT
SCHEMBL8736479 0.76 MAOB (0.63) PARP10PARP14MAPTCRHBPHTT
SCHEMBL25910322 0.75 MAPT (0.56) PARP10PARP14MAPTCRHBPHTT
SCHEMBL13257656 0.75 ALDH1A1 (0.76) PARP10PARP14MGLLHSD11B1
SCHEMBL25910319 0.74 MAOB (0.57) PARP10PARP14MAPTCRHBPHTT
SCHEMBL564525 0.73 RAB9A (0.70) PARP10PARP14MAPTCRHBPHTT
SCHEMBL4733674 0.72 ALDH1A1 (0.52) MAPTMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070020704-A1 Diaryl ureas with kinase inhibiting activity BAYER HEALTHCARE LLC 2007-01-25 US disclosed
US-20070020704-A1 Diaryl ureas with kinase inhibiting activity BAYER HEALTHCARE LLC 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070020704-A1 Diaryl ureas with kinase inhibiting activity FLT4, FLT1, FLT3 PARP10 1667/4885PARP14 2378/4885MAPT 2377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.