SCHEMBL14619954

SCHEMBL14619954

Cc1cc(C)c2c(c1)CC(C)N2

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CREBBP Q92793 7/20 0.37
BRD4 O60885 5/20 0.37
TSHR P16473 1/20 0.34
NNMT P40261 2/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
HSPA1A P0DMV8 1/20 0.31
PTPN7 P35236 1/20 0.31
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14256009 0.74 PNMT (0.49) TSHRKMT2AALDH1A1HSPA1AMAPT
SCHEMBL9791471 0.72 CREBBP (0.56) CREBBPBRD4TSHRKMT2AMEN1
SCHEMBL6028785 0.69 CREBBP (0.34) CREBBPBRD4TSHRNNMTKMT2A
SCHEMBL20023207 0.68 KDM4E (0.35) CREBBPTSHRNNMTKMT2AMEN1
SCHEMBL9336520 0.68 BRD4 (0.34) CREBBPBRD4NNMTKMT2AMEN1
SCHEMBL7922397 0.68 GAA (0.47) CREBBPBRD4TSHRALDH1A1HTR2A
SCHEMBL30101714 0.68 GAA (0.47) CREBBPBRD4TSHRALDH1A1HTR2A
SCHEMBL2266750 0.67 NNMT (0.34) CREBBPBRD4TSHRNNMT
SCHEMBL12965849 0.66 AR (0.45) CREBBPBRD4TSHRNNMTALDH1A1
SCHEMBL21729487 0.65 NNMT (0.58) TSHRNNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176312-B2 Kinase inhibitor scaffolds and methods for their preparation THE SCRIPPS RESEARCH INSTITUTE (US) 2007-02-13 US disclosed