SCHEMBL14635533

SCHEMBL14635533

Oc1nc2c(cc1F)CNCC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HTR2C P28335 3/20 0.36
HTR2B P41595 2/20 0.36
ADCY6 O43306 1/20 0.35
ADCY3 O60266 1/20 0.35
ADCY9 O60503 1/20 0.35
ADCY5 O95622 1/20 0.35
ADCY8 P40145 1/20 0.35
ADCY7 P51828 1/20 0.35
ADCY2 Q08462 1/20 0.35
ADCY1 Q08828 1/20 0.35
ADCY4 Q8NFM4 1/20 0.35
PNMT P11086 4/20 0.34
CD44 P16070 1/20 0.34
MAOB P27338 1/20 0.34
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14635622 0.81 CYP3A4 (0.44) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
SCHEMBL26959998 0.79 CYP3A4 (0.43) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
SCHEMBL31621544 0.78 CYP3A4 (0.40) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
Hydrochloric Acid SCHEMBL26914890 0.78 CYP3A4 (0.43) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
SCHEMBL24602646 0.78 CYP3A4 (0.40) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
Hydrochloric Acid SCHEMBL26631617 0.77 CYP3A4 (0.39) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
SCHEMBL29098326 0.75 CYP3A4 (0.37) CYP3A4POLBSMN1; SMN2HTR2CHTR2B
SCHEMBL6611519 0.70 CYP3A4 (0.47) CYP3A4POLBSMN1; SMN2HTR2CPNMT
SCHEMBL21465735 0.70 ADCY6 (0.57) ADCY6ADCY3ADCY9ADCY5ADCY8
SCHEMBL6607763 0.70 CYP3A4 (0.47) CYP3A4POLBSMN1; SMN2HTR2CPNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013010453-A1 CHEMOKING RECEPTOR ANTAGONISTS ABBOTT LABORATORIES (US) 2013-01-24 WO disclosed