Meradimate

Meradimate

SCHEMBL14637358

CC(C)[C@@H]1CC[C@@H](C)C[C@H]1OC(=O)c1ccccc1N.CC(C)[C@@H]1CC[C@@H](C)C[C@H]1OC(=O)c1ccccc1N

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 1.00
HPGD P15428 3/20 1.00
KDM4E B2RXH2 3/20 0.58
MAPT P10636 2/20 0.58
MAPK1 P28482 2/20 0.58
GAA P10253 1/20 0.58
ACLY P53396 1/20 0.53
LMNA P02545 2/20 0.51
NPSR1 Q6W5P4 3/20 0.50
CYP19A1 P11511 2/20 0.50
TSHR P16473 2/20 0.49
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
P2RX4 Q99571 1/20 0.47
EPHX1 P07099 2/20 0.46
POLB P06746 1/20 0.46
HSD17B10 Q99714 1/20 0.46
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
MITF O75030 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Meradimate SCHEMBL29461397 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL339007 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL14697604 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL18884 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL18989595 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL6851307 1.00 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL29209240 0.99 ALDH1A1 (0.98) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL8329573 0.99 ALDH1A1 (0.98) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL27915999 0.96 ALDH1A1 (0.93) ALDH1A1HPGDKDM4EMAPTMAPK1
Meradimate SCHEMBL19717873 0.95 ALDH1A1 (0.91) ALDH1A1HPGDKDM4EMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3523350-A1 ULTRAVIOLET RADIATION ABSORBING POLYMER COMPOSITION BASF SE (DE) 2019-08-14 EP disclosed
EP-3481365-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2019-05-15 EP disclosed
WO-2018065341-A1 ULTRAVIOLET RADIATION ABSORBING POLYMER COMPOSITION BASF SE (DE) 2018-04-12 WO disclosed
WO-2018007577-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2018-01-11 WO disclosed
EP-3229766-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2017-10-18 EP disclosed
EP-3191075-A1 MIXTURES OF COSMETIC UV ABSORBERS BASF SE (DE) 2017-07-19 EP disclosed
EP-3128993-A1 MIXTURES OF COSMETIC UV ABSORBERS BASF SE (DE) 2017-02-15 EP disclosed
EP-3128995-A1 SOLUBLIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2017-02-15 EP disclosed
EP-3041904-A1 STYRYL SULFIDE DYES BASF SE (DE) 2016-07-13 EP disclosed
WO-2016091930-A1 SOLUBILIZING AGENTS FOR UV FILTERS IN COSMETIC FORMULATIONS BASF SE (DE) 2016-06-16 WO disclosed
EP-2919773-A1 METHODS OF TREATMENT OF KERATINOCYTE-DERIVED LESIONS The Trustees of Columbia University in the City of New York (US) 2015-09-23 EP disclosed
WO-2015059368-A1 METHOD FOR DYEING KERATIN FIBRES USING CATIONIC STYRYL DISULPHIDE DYES, AND COMPOSITION INCLUDING SAID DYES L'OREAL (FR) 2015-04-30 WO disclosed
WO-2015028543-A1 STYRYL SULFIDE DYES BASF SE (DE) 2015-03-05 WO disclosed
EP-2744907-A1 METHOD FOR PRODUCING 4-AMINOBUTYRIC ACID FROM ALGAE Evonik Degussa GmbH (DE) 2014-06-25 EP disclosed
EP-2734180-A2 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION CONTAINING A MEROCYANINE DERIVATIVE COMPRISING SPECIFIC POLAR GROUPS CONSISTING OF HYDROXYL- AND ETHER-FUNCTIONALITIES L'OREAL (FR) 2014-05-28 EP disclosed
WO-2014078868-A1 METHODS OF TREATMENT OF KERATINOCYTE-DERIVED LESIONS THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2014-05-22 WO disclosed
EP-2709977-A2 USE OF BENZOTROPOLONE DERIVATIVES AS PHOTOSTABILIZER AND ANTIOXIDANT FOR STABILIZATION OF BODY-CARE AND HOUSEHOLD PRODUCTS. BASF SE (DE) 2014-03-26 EP disclosed
WO-2013023873-A1 METHOD FOR PRODUCING 4-AMINOBUTYRIC ACID FROM ALGAE EVONIK GOLDSCHMIDT GMBH (DE) 2013-02-21 WO disclosed
WO-2013010590-A1 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION CONTAINING A MEROCYANINE DERIVATIVE COMPRISING SPECIFIC POLAR GROUPS CONSISTING OF HYDROXYL- AND ETHER-FUNCTIONALITIES L'OREAL (FR) 2013-01-24 WO disclosed
WO-2013011094-A2 COSMETIC AND/OR DERMATOLOGICAL COMPOSITION CONTAINING A MEROCYANINE DERIVATIVE COMPRISING SPECIFIC POLAR GROUPS CONSISTING OF HYDROXYL- AND ETHER-FUNCTIONALITIES L'OREAL (FR) 2013-01-24 WO disclosed