SCHEMBL14637459

SCHEMBL14637459

CC1(C(=O)Nc2ccc([N+](=O)[O-])cc2)CCCNC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.53
NPSR1 Q6W5P4 2/20 0.53
HTR1E P28566 1/20 0.53
S1PR3 Q99500 1/20 0.53
HSPA9 P38646 2/20 0.49
MEN1 O00255 4/20 0.48
KMT2A Q03164 4/20 0.48
ALDH1A1 P00352 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
GAA P10253 2/20 0.45
LMNA P02545 4/20 0.45
NAMPT P43490 1/20 0.45
PTGES O14684 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
NPC1 O15118 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
EPHX1 P07099 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17729035 0.83 L3MBTL1 (0.43) NPSR1ALDH1A1L3MBTL1GAALMNA
Piperidine SCHEMBL27716285 0.74 KMT2A (0.62) MAPTMEN1KMT2AALDH1A1GAA
SCHEMBL10626089 0.71 MEN1 (0.57) MAPTNPSR1HTR1ES1PR3MEN1
Azetidine SCHEMBL27897562 0.70 ADRB1 (0.59) MAPTALDH1A1GAALMNATDP1
SCHEMBL18129842 0.69 CCR2 (0.33) KMT2AALDH1A1SMN1; SMN2KDM4ECYP3A4
SCHEMBL14637825 0.68 MAPK1 (0.38) MAPTNPSR1HTR1ES1PR3HSPA9
SCHEMBL642700 0.67 KMT2A (0.81) MAPTMEN1KMT2AALDH1A1GAA
SCHEMBL16922176 0.67 KMT2A (0.81) MAPTMEN1KMT2AALDH1A1GAA
SCHEMBL6302157 0.67 MEN1 (1.00) MAPTNPSR1MEN1KMT2AGAA
SCHEMBL1177730 0.67 MEN1 (1.00) MAPTNPSR1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013012827-A1 DIAMINOCYCLOHEXANE COMPOUNDS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-24 WO disclosed
WO-2013012829-A1 DIAMINOCYCLOHEXANE COMPOUNDS AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2013-01-24 WO disclosed