SCHEMBL14642116

SCHEMBL14642116

COc1ccc(OC)c(Sc2cc(-c3ccc(OCN)cc3C)nc(N)n2)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHFR P00374 5/20 0.42
LRRK2 Q5S007 4/20 0.39
TYMS P04818 2/20 0.39
EGFR P00533 1/20 0.39
KDR P35968 1/20 0.39
HSP90AA1 P07900 3/20 0.39
HSP90AB1 P08238 3/20 0.39
CHRNA7 P36544 1/20 0.39
TLR8 Q9NR97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4086287 0.89 DHFR (0.40) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4093637 0.89 MAOB (0.48) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4086671 0.88 DHFR (0.39) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4094840 0.88 DHFR (0.39) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4095647 0.88 MEN1 (0.39) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4093475 0.85 NPC1 (0.43) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4093485 0.85 DHFR (0.46) DHFRLRRK2TYMSEGFRKDR
SCHEMBL13927519 0.82 HSP90AA1 (0.48) DHFRLRRK2TYMSEGFRKDR
SCHEMBL4093607 0.81 DHFR (0.42) DHFRLRRK2TYMSEGFRKDR
SCHEMBL15101660 0.80 TSHR (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2036895-B1 HSP90 INHIBITOR CHUGAI PHARMACEUTICAL CO LTD (JP) 2013-01-16 EP disclosed