SCHEMBL14642940

SCHEMBL14642940

CCCCCCc1ccc(-c2ccc(CNCCCO[PH](=O)O)nc2-c2ccccc2)cc1CCC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 9/20 0.50
KDM4E B2RXH2 2/20 0.34
MEN1 O00255 1/20 0.34
APAF1 O14727 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ESR1 P03372 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CNR1 P21554 1/20 0.33
CNR2 P34972 1/20 0.33
SLC2A1 P11166 2/20 0.32
SOAT1 P35610 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL36170 0.84 S1PR3 (0.71) S1PR3
SCHEMBL2635044 0.83 S1PR3 (0.50) S1PR3KDM4EMEN1APAF1USP2
SCHEMBL14642685 0.80 S1PR3 (0.31) S1PR3
SCHEMBL35623 0.76 S1PR3 (0.59) S1PR3CNR1
SCHEMBL14642670 0.75 S1PR3 (0.46) S1PR3KDM4EMEN1ALDH1A1MAPT
SCHEMBL36218 0.73 S1PR3 (0.55) S1PR3
SCHEMBL13471220 0.72 SLC2A1 (0.47) S1PR3CNR1CNR2SLC2A1
SCHEMBL14642772 0.71 S1PR3 (0.40) S1PR3
SCHEMBL36337 0.70 S1PR3 (0.87) S1PR3
SCHEMBL13471216 0.70 DGAT2 (0.39) S1PR3KDM4ESLC2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130018019-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY ALLERGAN, INC. (US) 2013-01-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130018019-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY S1PR1, S1PR3, S1PR2 S1PR3 2/4885KDM4E 2618/4885MEN1 2735/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.