SCHEMBL2635044

SCHEMBL2635044

[CH2]CCNCc1ccc(-c2ccc(CCCCCC)c(CCC)c2)c(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 8/20 0.50
SOAT1 P35610 3/20 0.35
GPR84 Q9NQS5 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
APAF1 O14727 1/20 0.34
USP2 O75604 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ESR1 P03372 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
CACNA1B Q00975 1/20 0.34
APBA1 Q02410 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
TLR8 Q9NR97 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL36170 0.86 S1PR3 (0.71) S1PR3
SCHEMBL14642940 0.83 S1PR3 (0.50) S1PR3SOAT1KDM4EMEN1APAF1
SCHEMBL35623 0.77 S1PR3 (0.59) S1PR3
SCHEMBL36218 0.73 S1PR3 (0.55) S1PR3
SCHEMBL36337 0.70 S1PR3 (0.87) S1PR3
SCHEMBL2635686 0.69 S1PR3 (0.43) S1PR3KDM4EMEN1USP2ALDH1A1
SCHEMBL805669 0.67 S1PR3 (1.00) S1PR3
SCHEMBL13279803 0.66 S1PR1 (0.43) S1PR3
SCHEMBL13478408 0.64 GPR84 (0.44) SOAT1GPR84KDM4EALDH1A1
SCHEMBL10429729 0.63 LIPG (0.45) SOAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569322-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY Allergan, Inc. (US) 2013-03-20 EP disclosed
WO-2011143332-A1 AROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHONATE (S1P) RECEPTOR ACTIVITY ALLERGAN, INC. (US) 2011-11-17 WO disclosed