SCHEMBL14645495

SCHEMBL14645495

O=C(O)C1(I)CC1c1ccc(F)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.45
KDM1A O60341 3/20 0.41
RCOR1 Q9UKL0 3/20 0.41
PTGS2 P35354 1/20 0.41
HSD11B1 P28845 9/20 0.40
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
EPHX1 P07099 1/20 0.37
CCR2 P41597 1/20 0.36
MAPK1 P28482 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC9A1 P19634 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5266179 0.82 MAPK1 (0.49) KDM1AMAPK1CYP2C19
SCHEMBL28876302 0.76 LIG1 (0.44) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL17984248 0.76 KDM1A (0.44) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL28065197 0.76 KDM1A (0.44) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL16455153 0.76 KDM1A (0.44) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL19385670 0.74 LIG1 (0.41) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL19385671 0.74 LIG1 (0.41) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL4134830 0.74 KDM1A (0.41) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL5899615 0.73 KDM1A (0.44) LIG1KDM1ARCOR1PTGS2HSD11B1
SCHEMBL15797670 0.71 KDM1A (0.44) KDM1ARCOR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729447-A1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H. Lundbeck A/S (DK) 2014-05-14 EP disclosed
WO-2013007621-A1 POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR H. LUNDBECK A/S (DK) 2013-01-17 WO disclosed