SCHEMBL14645980

SCHEMBL14645980

CCCCC(Cc1c(C#N)cc(C(=O)O)c(N)c1C)c1c(C#N)cc(C(=O)O)c(N)c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.35
HPGD P15428 3/20 0.35
ADRB2 P07550 1/20 0.34
KDM4E B2RXH2 5/20 0.33
POLB P06746 2/20 0.33
HSD17B10 Q99714 2/20 0.33
TSHR P16473 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
BRS3 P32247 1/20 0.32
LMNA P02545 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GABRP O00591 1/20 0.30
GABRD O14764 1/20 0.30
GABRA1 P14867 1/20 0.30
GABRB1 P18505 1/20 0.30
GABRG2 P18507 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14645957 0.81 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL14645997 0.81 ALDH1A1 (0.43) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL14645962 0.78 KDM4E (0.42) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL14645817 0.76 KDM4E (0.42) ALDH1A1KDM4EPOLBHSD17B10L3MBTL1
SCHEMBL10769054 0.72 KDM4E (0.38) ALDH1A1KDM4ETSHRL3MBTL1BRS3
SCHEMBL14645847 0.70 KDM4E (0.46) KDM4EHSD17B10L3MBTL1TDP1GABRP
SCHEMBL14645991 0.70 HTT (0.44) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL2535736 0.67 KDM4E (0.38) ALDH1A1KDM4EPOLBTSHRL3MBTL1
SCHEMBL12474718 0.65 KDM4E (0.42) ALDH1A1HPGDKDM4EHSD17B10BRS3
SCHEMBL3221189 0.64 ALDH1A1 (0.34) ALDH1A1KDM4ETSHRL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729444-B1 METHOD FOR MANUFACTURING 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE BAYER IP GMBH (DE) 2017-08-23 EP disclosed
EP-2729444-A1 METHOD FOR THE PRODUCTION OF 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE Bayer Intellectual Property GmbH (DE) 2014-05-14 EP disclosed
WO-2013007603-A1 METHOD FOR THE PRODUCTION OF 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-01-17 WO disclosed