SCHEMBL14645997

SCHEMBL14645997

CCCCCCc1c(C#N)cc(C(=O)O)c(N)c1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
KAT8 Q9H7Z6 2/20 0.42
PPARA Q07869 2/20 0.42
RARB P10826 3/20 0.41
CSNK2B P67870 2/20 0.40
CSNK2A1 P68400 2/20 0.40
PIP5K1A Q99755 1/20 0.40
PPARG P37231 1/20 0.39
KDM4E B2RXH2 2/20 0.39
HSD17B10 Q99714 2/20 0.39
RARA P10276 1/20 0.39
RARG P13631 1/20 0.39
POLB P06746 1/20 0.38
TSHR P16473 1/20 0.38
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14645957 1.00 ALDH1A1 (0.43) ALDH1A1HPGDKAT8PPARARARB
SCHEMBL14645817 0.90 KDM4E (0.42) ALDH1A1KDM4EHSD17B10POLB
SCHEMBL14645962 0.86 KDM4E (0.42) ALDH1A1HPGDKDM4EHSD17B10TSHR
SCHEMBL14645980 0.81 ALDH1A1 (0.35) ALDH1A1HPGDCSNK2BCSNK2A1PIP5K1A
SCHEMBL14645847 0.78 KDM4E (0.46) KDM4EHSD17B10GABRPGABRDGABRA1
SCHEMBL14645991 0.77 HTT (0.44) ALDH1A1HPGDKDM4EHSD17B10POLB
SCHEMBL30061109 0.77 RARB (0.48) KAT8PPARARARBPPARGKDM4E
SCHEMBL578085 0.77 RARB (0.48) KAT8PPARARARBPPARGKDM4E
SCHEMBL8770841 0.77 GABRP (0.48) KAT8PPARARARBPPARGKDM4E
SCHEMBL7744473 0.76 RARB (0.46) KAT8PPARARARBPPARGKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729444-B1 METHOD FOR MANUFACTURING 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE BAYER IP GMBH (DE) 2017-08-23 EP disclosed
EP-2729444-A1 METHOD FOR THE PRODUCTION OF 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE Bayer Intellectual Property GmbH (DE) 2014-05-14 EP disclosed
WO-2013007603-A1 METHOD FOR THE PRODUCTION OF 2-AMINO-5-CYANO-N,3-DIMETHYLBENZAMIDE BAYER INTELLECTUAL PROPERTY GMBH (DE) 2013-01-17 WO disclosed