SCHEMBL14686017

SCHEMBL14686017

CCCc1n[nH]c2c(=O)[nH]c(Cc3cc(S(=O)(=O)NC(=O)c4ccc(C(C)(C)C)cc4)ccc3OCC)nc12

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.39
PDE5A O76074 18/20 0.38
HDAC1 Q13547 9/20 0.38
HDAC6 Q9UBN7 9/20 0.38
HDAC2 Q92769 8/20 0.38
HDAC3 O15379 2/20 0.38
NCOR2 Q9Y618 2/20 0.38
PTPN1 P18031 1/20 0.36
PDE2A O00408 1/20 0.35
PDE9A O76083 1/20 0.35
PDE4A P27815 1/20 0.35
PDE6C P51160 1/20 0.35
PDE1A P54750 1/20 0.35
PDE11A Q9HCR9 1/20 0.35
PDE10A Q9Y233 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14685955 0.86 KDM4E (0.41) KDM4EPDE5AHDAC1HDAC6HDAC2
SCHEMBL14686005 0.86 PDE5A (0.39) KDM4EPDE5AHDAC1HDAC6HDAC2
SCHEMBL14686015 0.80 KDM4E (0.45) KDM4EPDE5AHDAC1HDAC6HDAC2
SCHEMBL3671939 0.76 PDE5A (0.55) PDE5APDE2APDE9APDE4APDE6C
SCHEMBL17333641 0.74 PDE5A (0.47) KDM4EPDE5AHDAC1HDAC6HDAC2
SCHEMBL5988676 0.74 PDE5A (0.48) PDE5AHDAC1HDAC6HDAC2PDE2A
SCHEMBL16972452 0.74 PDE1A (0.48) KDM4EPDE5APDE2APDE9APDE4A
SCHEMBL5085823 0.73 PDE5A (0.56) PDE5AHDAC1HDAC6HDAC2HDAC3
SCHEMBL7002705 0.72 KDM4E (0.73) KDM4EPDE5AHDAC1HDAC6HDAC2
SCHEMBL7007807 0.72 KDM4E (0.61) KDM4EPDE5AHDAC1HDAC6HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2556820-A2 COMPOSITION CONTAINING PDE5 INHIBITOR FOR RELIEVING SKIN WRINKLES SK Chemicals, Co., Ltd. (KR) 2013-02-13 EP disclosed