SCHEMBL14686396

SCHEMBL14686396

CS(=O)(=O)[CH]c1cccnc1OC(F)F

nearest known ligand 0.54

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.54
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NFE2L2 Q16236 9/20 0.36
LPAR1 Q92633 2/20 0.33
SLC22A12 Q96S37 1/20 0.33
TYK2 P29597 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
DRD1 P21728 2/20 0.32
TRIM24 O15164 1/20 0.31
TRIM33 Q9UPN9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16114579 0.79 TRPV4 (0.53) TRPV4NR3C1PGRLPAR1DRD1
SCHEMBL14686369 0.76 TRPV4 (0.43) TRPV4NR3C1PGRNFE2L2DRD1
SCHEMBL14686367 0.74 L3MBTL1 (0.46) SLC22A12DRD1
SCHEMBL2376210 0.73 TRPV4 (0.54) TRPV4NR3C1PGRLPAR1TYK2
SCHEMBL31328368 0.71 TRPV4 (0.51) TRPV4NR3C1PGRLPAR1TYK2
SCHEMBL22679340 0.70 TRPV4 (0.50) TRPV4NR3C1PGRLPAR1TYK2
SCHEMBL21144313 0.70 TRPV4 (1.00) TRPV4NR3C1PGRNFE2L2SLC22A12
SCHEMBL14686293 0.70 PTGS1 (0.34) TRPV4NFE2L2
SCHEMBL14686399 0.70 CA12 (0.36) TRPV4NFE2L2
SCHEMBL2646025 0.70 TRPV4 (0.57) TRPV4NR3C1PGRLPAR1TYK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1865940-B1 ALPHA KETOAMIDE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-02-13 EP claimed