SCHEMBL14686293

SCHEMBL14686293

CS(=O)(=O)[CH]c1ccncc1OC(F)F

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 7/20 0.34
PTGS2 P35354 7/20 0.34
CA12 O43570 3/20 0.33
CA2 P00918 3/20 0.33
CA9 Q16790 3/20 0.33
CA1 P00915 2/20 0.33
GAA P10253 1/20 0.33
CA14 Q9ULX7 2/20 0.32
CYP17A1 P05093 1/20 0.32
NAMPT P43490 1/20 0.31
TRPV4 Q9HBA0 1/20 0.31
BACE1 P56817 1/20 0.31
NFE2L2 Q16236 1/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14686399 0.88 CA12 (0.36) PTGS1PTGS2CA12CA2CA9
SCHEMBL14686367 0.78 L3MBTL1 (0.46) CA12CA2CA9CA1GAA
SCHEMBL2377439 0.73 LMNA (0.34) PTGS1PTGS2CA12CA2CA9
SCHEMBL14686369 0.70 TRPV4 (0.43) TRPV4NFE2L2
SCHEMBL2378342 0.70 CA12 (0.37) PTGS1PTGS2CA12CA2CA9
SCHEMBL14686396 0.70 TRPV4 (0.54) TRPV4NFE2L2
SCHEMBL16114581 0.69 DRD1 (0.38) CA12CA2CA9GAACA14
SCHEMBL14943109 0.69 CYP2E1 (0.38) CA12CA2CA9CA1GAA
SCHEMBL28038210 0.68 SLC22A12 (0.41) PTGS1PTGS2CYP17A1
SCHEMBL31543981 0.68 KDM4E (0.37) GAATRPV4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1865940-B1 ALPHA KETOAMIDE COMPOUNDS AS CYSTEINE PROTEASE INHIBITORS VIROBAY INC (US) 2013-02-13 EP claimed