SCHEMBL14690797

SCHEMBL14690797

CC(C)(C)[Si](C)(C)OCCCCC1CNC(=O)O1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DUT P33316 2/20 0.39
LMNA P02545 2/20 0.39
MAOA P21397 1/20 0.39
SLC6A2 P23975 1/20 0.39
PKM P14618 1/20 0.38
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
MAPK1 P28482 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SYK P43405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14690796 1.00 DUT (0.39) DUTLMNAMAOASLC6A2PKM
SCHEMBL21400915 0.96 DUT (0.40) DUTLMNAMAOASLC6A2PKM
SCHEMBL16180004 0.91 LMNA (0.40) DUTLMNAMAOASLC6A2PKM
SCHEMBL2287916 0.91 LMNA (0.40) DUTLMNAMAOASLC6A2PKM
SCHEMBL1712032 0.91 LMNA (0.40) DUTLMNAMAOASLC6A2PKM
SCHEMBL21428625 0.82 LMNA (0.49) LMNAMAOASLC6A2PKMUSP2
SCHEMBL2288476 0.82 LMNA (0.49) LMNAMAOASLC6A2PKMUSP2
SCHEMBL20519513 0.82 LMNA (0.49) LMNAMAOASLC6A2PKMUSP2
SCHEMBL591257 0.75 ALDH1A1 (0.44) DUTALDH1A1MAPK1
SCHEMBL16878814 0.73 DUT (0.36) DUT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8916573-B2 Quinazoline-2,4-dione derivatives ACTELION PHARMACEUTICALS LTD. (CH) 2014-12-23 US disclosed
US-20140171425-A1 QUINAZOLINE-2,4-DIONE DERIVATIVES ACTELION PHARMACEUTICALS LTD. (CH) 2014-06-19 US disclosed
EP-2742042-A1 QUINAZOLINE-2,4-DIONE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2014-06-18 EP disclosed
WO-2013021363-A1 QUINAZOLINE-2,4-DIONE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2013-02-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140171425-A1 QUINAZOLINE-2,4-DIONE DERIVATIVES NQO2, H1-3, H1-0 DUT 836/4885LMNA 2400/4885MAOA 1561/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.