SCHEMBL14693166

SCHEMBL14693166

CCNC(=O)Nc1ccc(Oc2ccnc3cc(OC[C@H](O)CN(CC)CC)c(C(=O)NC)cc23)cc1CI

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.40
MET P08581 6/20 0.40
AURKB Q96GD4 6/20 0.40
LCK P06239 5/20 0.40
AURKA O14965 4/20 0.40
TEK Q02763 4/20 0.40
AXL P30530 5/20 0.40
PDGFRA P16234 9/20 0.38
KIT P10721 4/20 0.38
FGFR2 P21802 4/20 0.38
FLT1 P17948 5/20 0.37
FLT4 P35916 5/20 0.37
RIPK2 O43353 4/20 0.37
RET P07949 4/20 0.37
PDGFRB P09619 4/20 0.37
DDR1 Q08345 4/20 0.37
DDR2 Q16832 4/20 0.37
FGFR1 P11362 4/20 0.37
STK10 O94804 3/20 0.37
ABL1 P00519 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14693181 0.96 KDR (0.45) KDRMETAURKBLCKAURKA
SCHEMBL14693173 0.95 KDR (0.41) KDRMETAURKBLCKAURKA
SCHEMBL14693175 0.94 KDR (0.43) KDRMETAURKBLCKAURKA
SCHEMBL12673525 0.91 KDR (0.46) KDRMETAURKBLCKAURKA
SCHEMBL1248445 0.90 KDR (0.48) KDRMETAURKBLCKAURKA
SCHEMBL1248449 0.90 KDR (0.48) KDRMETAURKBLCKAURKA
SCHEMBL14693152 0.88 MET (0.39) KDRMETAURKBLCKAURKA
SCHEMBL14693180 0.87 FGFR2 (0.46) KDRMETAURKBLCKAURKA
SCHEMBL14437505 0.86 AXL (0.52) KDRMETAURKBLCKAURKA
SCHEMBL12673816 0.86 KDR (0.47) KDRMETAURKBLCKAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8372981-B2 Nitrogen-containing aromatic derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2013-02-12 US disclosed