SCHEMBL14701619

SCHEMBL14701619

C#CCOc1ccc(CN(CCCCCC(=O)O)Cc2nccn2CC(=O)N(CC(N)=O)CC(=O)O)cc1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.34
PPARA Q07869 3/20 0.34
GABRA1 P14867 1/20 0.34
GABRB2 P47870 1/20 0.34
CXCR4 P61073 1/20 0.33
ALOX5 P09917 1/20 0.33
CYP19A1 P11511 1/20 0.33
FFAR1 O14842 1/20 0.31
FFAR4 Q5NUL3 1/20 0.31
HDAC3 O15379 1/20 0.30
HDAC2 Q92769 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
NCOR2 Q9Y618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14674656 0.87 PPARG (0.33) PPARGPPARAGABRA1GABRB2CXCR4
SCHEMBL14674855 0.82 GABRA1 (0.35) PPARGPPARAGABRA1GABRB2CXCR4
SCHEMBL16374660 0.74 CXCR4 (0.33) PPARGPPARACXCR4ALOX5HDAC3
SCHEMBL15199009 0.73 CA1 (0.44)
SCHEMBL2834770 0.73 TBXAS1 (0.31) CXCR4
SCHEMBL15197274 0.72 PPARG (0.33) PPARGPPARAHDAC3HDAC2HDAC8
SCHEMBL14674925 0.71 FOLH1 (0.34)
SCHEMBL15198937 0.69 CA1 (0.52)
SCHEMBL15198936 0.69 CA1 (0.46)
SCHEMBL16374705 0.68 FPR2 (0.35) CXCR4HDAC3HDAC2HDAC8NCOR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013022797-A1 RADIOLABELED PROSTATE SPECIFIC MEMBRANE ANTIGEN INHIBITORS MOLECULAR INSIGHT PHARMACEUTICALS (US) 2013-02-14 WO disclosed