SCHEMBL14715396

SCHEMBL14715396

COc1cc2nc(N3CCC(Cc4ccccc4)(OC(=O)NCc4ccc(Cl)c(Cl)c4)CC3)nc(N)c2cc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 4/20 0.50
ADRA1B P35368 4/20 0.50
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 1/20 0.47
NPC1 O15118 1/20 0.47
SLC22A2 O15244 1/20 0.47
SLC22A1 O15245 1/20 0.47
ABCC4 O15439 1/20 0.47
SLC22A3 O75751 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
MMP1 P03956 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47
GLA P06280 1/20 0.47
CHRM2 P08172 1/20 0.47
CYP3A4 P08684 1/20 0.47
HTR1A P08908 1/20 0.47
ADRA2A P08913 1/20 0.47
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715262 0.92 ADRA1A (0.56) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL14715306 0.90 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL3319263 0.89 ADRA1A (0.52) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL14715408 0.88 ADRA1A (0.50) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL14715512 0.87 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL14715477 0.86 ADRA1A (0.49) ADRA1AADRA1B
SCHEMBL14715409 0.85 ADRA1A (0.57) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL14715297 0.84 ADRA1A (0.54) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL2187625 0.84 ADRA1A (0.47) ADRA1AADRA1BKDM4EMEN1NPC1
SCHEMBL2172942 0.84 ADRA1A (0.47) ADRA1AADRA1BKDM4EMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed