SCHEMBL14715409

SCHEMBL14715409

COc1cc2nc(N3CCC(Cc4ccccc4)(OC(=O)NCc4ccco4)CC3)nc(N)c2cc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 7/20 0.57
ADRA1B P35368 7/20 0.57
KDM4E B2RXH2 3/20 0.57
GLA P06280 3/20 0.57
GAA P10253 3/20 0.57
ADRA1D P25100 3/20 0.57
ALDH1A1 P00352 2/20 0.57
LMNA P02545 2/20 0.57
CYP3A4 P08684 2/20 0.57
MAPT P10636 2/20 0.57
HPGD P15428 2/20 0.57
ADRA2B P18089 2/20 0.57
ADRA2C P18825 2/20 0.57
OPRM1 P35372 2/20 0.57
HSD17B10 Q99714 2/20 0.57
MEN1 O00255 1/20 0.57
NPC1 O15118 1/20 0.57
SLC22A2 O15244 1/20 0.57
SLC22A1 O15245 1/20 0.57
ABCC4 O15439 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715262 0.91 ADRA1A (0.56) ADRA1AADRA1BKDM4EGLAGAA
SCHEMBL2174205 0.89 ADRA1A (0.59) ADRA1AADRA1BKDM4EGLAGAA
SCHEMBL14715306 0.87 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL14715512 0.86 ADRA1A (0.51) ADRA1AADRA1B
SCHEMBL14715396 0.85 ADRA1A (0.50) ADRA1AADRA1BKDM4EGLAGAA
SCHEMBL14715408 0.85 ADRA1A (0.50) ADRA1AADRA1BKDM4EGLAGAA
SCHEMBL14715477 0.83 ADRA1A (0.49) ADRA1AADRA1B
SCHEMBL14715297 0.82 ADRA1A (0.54) ADRA1AADRA1BKDM4EGLAGAA
SCHEMBL14715376 0.82 WHR1 (0.46) ADRA1AADRA1B
SCHEMBL14715455 0.82 ADRA1A (0.55) ADRA1AADRA1BGLAADRA1DCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed