SCHEMBL14715436

SCHEMBL14715436

COc1cc2nc(N3CCC(CC4CCC4)(OC(=O)NC4CCc5ccccc5C4)CC3)nc(O)c2cc1OC

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
WHR1 P49842 2/20 0.42
ADRA1B P35368 6/20 0.40
ADRA1A P35348 4/20 0.40
ADRA1D P25100 4/20 0.40
EHMT2 Q96KQ7 4/20 0.39
ADRA2A P08913 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715370 0.89 EHMT2 (0.44) ADRA1BADRA1AEHMT2
SCHEMBL2171720 0.88 WHR1 (0.42) WHR1ADRA1BADRA1AADRA1DEHMT2
SCHEMBL14715446 0.88 WHR1 (0.49) WHR1ADRA1BADRA1AADRA1DEHMT2
SCHEMBL13333113 0.85 ADRA1A (0.43) WHR1ADRA1BADRA1AADRA1DEHMT2
SCHEMBL2170814 0.84 WHR1 (0.45) WHR1ADRA1BADRA1AADRA1DEHMT2
SCHEMBL14715393 0.84 EHMT2 (0.45) WHR1ADRA1BADRA1AEHMT2
SCHEMBL14715357 0.83 EHMT2 (0.45) WHR1EHMT2
SCHEMBL14715170 0.82 ADRA1A (0.51) ADRA1BADRA1AADRA1D
SCHEMBL13333129 0.81 ADRA1A (0.45) WHR1ADRA1BADRA1AADRA1DEHMT2
SCHEMBL7919688 0.80 EHMT2 (0.45) ADRA1BADRA1AEHMT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed