SCHEMBL14715446

SCHEMBL14715446

COc1cc2nc(N3CCC(CC4CCC4)(OC(=O)NC4CCCC4)CC3)nc(O)c2cc1OC

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
WHR1 P49842 1/20 0.49
EHMT2 Q96KQ7 5/20 0.46
CCR4 P51679 10/20 0.45
ADRA2A P08913 1/20 0.42
ADRA2B P18089 1/20 0.42
ADRA2C P18825 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715436 0.88 WHR1 (0.42) WHR1EHMT2ADRA2AADRA2BADRA2C
SCHEMBL2171214 0.86 WHR1 (0.50) WHR1EHMT2CCR4ADRA2AADRA2B
SCHEMBL14715407 0.86 EHMT2 (0.48) WHR1EHMT2ADRA1DADRA1AADRA1B
SCHEMBL14715357 0.85 EHMT2 (0.45) WHR1EHMT2
SCHEMBL14715363 0.81 EHMT2 (0.44) WHR1EHMT2ADRA2AADRA2BADRA2C
SCHEMBL2170933 0.81 WHR1 (0.50) WHR1EHMT2ADRA2AADRA2BADRA2C
SCHEMBL14715415 0.80 EHMT2 (0.43) WHR1EHMT2
SCHEMBL14715448 0.79 ADRA2A (0.47) WHR1EHMT2ADRA2AADRA2BADRA2C
SCHEMBL2170814 0.78 WHR1 (0.45) WHR1EHMT2ADRA2AADRA2BADRA2C
SCHEMBL14715393 0.78 EHMT2 (0.45) WHR1EHMT2ADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed