SCHEMBL14715599

SCHEMBL14715599

O=C(N[C@H]1CC[C@H](CCN2CCC(Oc3ccc(F)cc3Cl)CC2)CC1)Oc1ccnc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.51
DRD2 P14416 13/20 0.48
DRD3 P35462 11/20 0.48
HTR2A P28223 10/20 0.48
HTR1A P08908 6/20 0.48
DRD4 P21917 3/20 0.48
HTR2C P28335 3/20 0.48
HTR2B P41595 3/20 0.48
DRD1 P21728 1/20 0.45
IDO1 P14902 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715677 0.92 AR (0.52) ARDRD2DRD3HTR2AHTR1A
SCHEMBL3087616 0.89 DRD3 (0.61) ARDRD2DRD3HTR2AHTR1A
SCHEMBL14715648 0.89 DRD2 (0.44) ARDRD2DRD3HTR2AHTR1A
SCHEMBL14715723 0.89 DRD2 (0.44) ARDRD2DRD3HTR2AHTR1A
SCHEMBL14715633 0.88 AR (0.48) ARDRD2DRD3HTR2AHTR1A
SCHEMBL14715628 0.86 DRD2 (0.49) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL14715630 0.84 DRD2 (0.51) ARDRD2DRD3HTR2AHTR1A
SCHEMBL14715692 0.83 DRD2 (0.49) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL3086163 0.81 DRD3 (0.59) ARDRD2DRD3HTR2AHTR1A
SCHEMBL27882701 0.81 HRH1 (0.47) DRD3HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed