SCHEMBL14715633

SCHEMBL14715633

O=C(N[C@H]1CC[C@H](CCN2CCC(Oc3ccc(F)cc3)CC2)CC1)Oc1ccnc2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.48
DRD2 P14416 14/20 0.48
HTR2A P28223 12/20 0.48
DRD3 P35462 12/20 0.48
HTR1A P08908 7/20 0.48
DRD4 P21917 3/20 0.46
HTR2C P28335 3/20 0.46
HTR2B P41595 3/20 0.46
TNKS O95271 1/20 0.44
DRD1 P21728 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715692 0.92 DRD2 (0.49) DRD2HTR2ADRD3HTR1ADRD4
SCHEMBL14715677 0.90 AR (0.52) ARDRD2HTR2ADRD3HTR1A
SCHEMBL14715599 0.88 AR (0.51) ARDRD2HTR2ADRD3HTR1A
SCHEMBL14715628 0.88 DRD2 (0.49) DRD2HTR2ADRD3HTR1ADRD4
SCHEMBL3083219 0.88 DRD3 (0.62) DRD2HTR2ADRD3HTR1ADRD4
SCHEMBL14715630 0.85 DRD2 (0.51) ARDRD2HTR2ADRD3HTR1A
SCHEMBL3073465 0.79 DRD3 (0.64) DRD2HTR2ADRD3HTR1ADRD4
SCHEMBL14715648 0.79 DRD2 (0.44) ARDRD2HTR2ADRD3HTR1A
SCHEMBL14715723 0.79 DRD2 (0.44) ARDRD2HTR2ADRD3HTR1A
SCHEMBL3086163 0.78 DRD3 (0.59) ARDRD2HTR2ADRD3HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed