SCHEMBL14715692

SCHEMBL14715692

O=C(N[C@H]1CC[C@H](CCN2CCC(Oc3ccncc3)CC2)CC1)Oc1ccnc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 16/20 0.49
DRD3 P35462 14/20 0.49
HTR2A P28223 11/20 0.49
HTR1A P08908 6/20 0.47
DRD4 P21917 3/20 0.47
HTR2C P28335 3/20 0.47
HTR2B P41595 3/20 0.47
NAMPT P43490 1/20 0.46
DRD1 P21728 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715633 0.92 AR (0.48) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL14715628 0.88 DRD2 (0.49) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL3073465 0.87 DRD3 (0.64) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL14715630 0.85 DRD2 (0.51) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL14715677 0.85 AR (0.52) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL14715599 0.83 AR (0.51) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL3083219 0.79 DRD3 (0.62) DRD2DRD3HTR2AHTR1ADRD4
SCHEMBL15911282 0.78 DRD2 (0.77) DRD2DRD3HTR2AHTR1A
SCHEMBL15911212 0.76 DRD2 (0.78) DRD2DRD3HTR2A
SCHEMBL3089494 0.76 DRD3 (0.64) DRD2DRD3HTR2AHTR1ADRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed