SCHEMBL14715696

SCHEMBL14715696

N#Cc1cc(Cl)ccc1OC1CCN(CC[C@H]2CC[C@H](C(N)=O)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.47
PROKR1 Q8TCW9 2/20 0.47
EPHX2 P34913 1/20 0.44
ALDH1A1 P00352 2/20 0.42
POLB P06746 1/20 0.42
TBK1 Q9UHD2 1/20 0.41
GAA P10253 1/20 0.41
HRH1 P35367 3/20 0.41
HTR2A P28223 3/20 0.41
DRD3 P35462 3/20 0.41
CCR3 P51677 2/20 0.41
KCNH2 Q12809 2/20 0.41
CHRM4 P08173 1/20 0.39
CHEK1 O14757 1/20 0.39
CHRM5 P08912 1/20 0.39
ADRA2A P08913 1/20 0.39
CYP2D6 P10635 1/20 0.39
DRD2 P14416 1/20 0.39
ADRA2B P18089 1/20 0.39
ADRA2C P18825 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3960275 1.00 FPR2 (0.47) FPR2PROKR1EPHX2ALDH1A1POLB
SCHEMBL3965016 0.91 FPR2 (0.46) FPR2PROKR1EPHX2TBK1HRH1
SCHEMBL3079707 0.88 HRH1 (0.44) ALDH1A1HRH1DRD3CCR3KCNH2
SCHEMBL14715627 0.88 HRH1 (0.44) ALDH1A1HRH1DRD3CCR3KCNH2
SCHEMBL3084815 0.88 DRD3 (0.52) FPR2PROKR1EPHX2HTR2ADRD3
SCHEMBL3960280 0.88 FPR2 (0.47) FPR2PROKR1EPHX2TBK1HRH1
SCHEMBL14715698 0.88 FPR2 (0.47) FPR2PROKR1EPHX2TBK1HRH1
Hydrochloric Acid SCHEMBL3074546 0.87 FPR2 (0.46) FPR2PROKR1EPHX2TBK1HRH1
SCHEMBL3959472 0.87 MEN1 (0.46) EPHX2ALDH1A1HTR2ADRD3KCNH2
Hydrochloric Acid SCHEMBL3074547 0.87 FPR2 (0.46) FPR2PROKR1EPHX2TBK1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed