SCHEMBL14715698

SCHEMBL14715698

N#Cc1cc(Cl)ccc1OC1CCN(CC[C@H]2CC[C@H](N)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FPR2 P25090 2/20 0.47
PROKR1 Q8TCW9 2/20 0.47
DRD2 P14416 1/20 0.41
EPHX2 P34913 1/20 0.41
NOS3 P29474 7/20 0.41
NOS1 P29475 7/20 0.41
NOS2 P35228 7/20 0.41
TBK1 Q9UHD2 2/20 0.40
HTR2A P28223 1/20 0.37
DRD3 P35462 1/20 0.37
HRH1 P35367 1/20 0.37
CCR3 P51677 1/20 0.37
KCNH2 Q12809 1/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
HRH3 Q9Y5N1 1/20 0.37
SLC6A4 P31645 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3960280 1.00 FPR2 (0.47) FPR2PROKR1DRD2EPHX2NOS3
Hydrochloric Acid SCHEMBL3074547 0.99 FPR2 (0.46) FPR2PROKR1DRD2EPHX2NOS3
Hydrochloric Acid SCHEMBL3074546 0.99 FPR2 (0.46) FPR2PROKR1DRD2EPHX2NOS3
SCHEMBL3960275 0.88 FPR2 (0.47) FPR2PROKR1DRD2EPHX2NOS3
SCHEMBL14715696 0.88 FPR2 (0.47) FPR2PROKR1DRD2EPHX2NOS3
SCHEMBL3087873 0.87 HRH1 (0.41) DRD2TBK1HRH1CCR3KCNH2
SCHEMBL3079710 0.87 HRH1 (0.41) DRD2TBK1HRH1CCR3KCNH2
SCHEMBL3965016 0.87 FPR2 (0.46) FPR2PROKR1EPHX2NOS3NOS1
SCHEMBL14715640 0.84 MEN1 (0.43) DRD2EPHX2HTR2ADRD3HRH1
SCHEMBL14715616 0.84 MEN1 (0.43) DRD2EPHX2HTR2ADRD3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed