SCHEMBL14715736

SCHEMBL14715736

N[C@H]1CC[C@H](CCN2CCC(Oc3ccc(Cl)c(Cl)c3)CC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 17/20 0.50
CCR3 P51677 17/20 0.50
KDM4E B2RXH2 1/20 0.49
KCNH2 Q12809 11/20 0.48
DRD2 P14416 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14715703 1.00 HRH1 (0.50) HRH1CCR3KDM4EKCNH2DRD2
SCHEMBL14715735 0.85 CCR3 (0.54) HRH1CCR3KCNH2
SCHEMBL3965013 0.85 CCR3 (0.54) HRH1CCR3KCNH2
SCHEMBL5369447 0.82 HRH1 (0.56) HRH1CCR3KDM4EKCNH2
SCHEMBL3067858 0.81 HTR7 (0.46) DRD2
SCHEMBL3067860 0.81 HTR7 (0.46) DRD2
SCHEMBL2923912 0.80 HRH1 (0.52) HRH1CCR3KDM4EKCNH2
SCHEMBL14715741 0.80 DRD2 (0.59) HRH1KCNH2DRD2
SCHEMBL5102799 0.80 HRH1 (0.59) HRH1CCR3KDM4EKCNH2
SCHEMBL3085004 0.79 NAMPT (0.52) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed