SCHEMBL14715744

SCHEMBL14715744

N#Cc1ccc(OC2CCN(CC[C@H]3CC[C@H](N)CC3)CC2)c(F)c1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.44
HRH2 P25021 1/20 0.42
HRH1 P35367 1/20 0.42
GPR6 P46095 15/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3075391 1.00 HRH3 (0.44) HRH3HRH2HRH1GPR6
SCHEMBL3959409 0.88 GPR6 (0.44) GPR6
SCHEMBL14715699 0.85 GRM2 (0.47) HRH3HRH1GPR6
SCHEMBL3086252 0.85 GRM2 (0.47) HRH3HRH1GPR6
SCHEMBL3087873 0.83 HRH1 (0.41) HRH3HRH1GPR6
SCHEMBL3079710 0.83 HRH1 (0.41) HRH3HRH1GPR6
SCHEMBL3963647 0.82 DRD2 (0.39) HRH3
SCHEMBL3087227 0.82 DRD2 (0.39) HRH3
SCHEMBL4233991 0.80 HRH3 (0.56) HRH3HRH1GPR6
SCHEMBL3960280 0.79 FPR2 (0.47) HRH3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079693-B1 ETHER DERIVATIVES DUAL MODULATORS OF THE 5-HT2A AND D3 RECEPTORS HOFFMANN LA ROCHE (CH) 2013-02-27 EP claimed