SCHEMBL14716928

SCHEMBL14716928

CNCCNC.CNCCNC

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 3/20 0.47
PRMT6 Q96LA8 3/20 0.47
PRMT8 Q9NR22 3/20 0.47
PRMT1 Q99873 2/20 0.47
PRMT3 O60678 1/20 0.47
EPHX1 P07099 1/20 0.44
TAAR1 Q96RJ0 4/20 0.35
ATM Q13315 1/20 0.35
HTR2A P28223 1/20 0.32
HRH1 P35367 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5425 1.00
SCHEMBL30273045 0.94 CARM1 (0.44) CARM1PRMT6PRMT8PRMT1PRMT3
SCHEMBL31327263 0.94
SCHEMBL29755267 0.94
Bromide SCHEMBL7115005 0.94
Ammonia Solution, Strong SCHEMBL2487756 0.94
SCHEMBL1393802 0.94
Iodide SCHEMBL7118709 0.94
Ammonia Solution, Strong SCHEMBL734851 0.94
SCHEMBL31726679 0.94

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9018382-B2 Indazoles GLAXOSMITHKLINE LLC (US) 2015-04-28 US disclosed
EP-2566328-B1 INDAZOLES GLAXOSMITHKLINE LLC (US) 2015-03-04 EP disclosed
US-20140350013-A1 INDAZOLES GLAXOSMITHKLINE LLC 2014-11-27 US disclosed
US-8846935-B2 Indazoles GLAXOSMITHKLINE LLC (US) 2014-09-30 US disclosed
US-20130053383-A1 INDAZOLES GLAXOSMITHKLINE LLC 2013-02-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130053383-A1 INDAZOLES IDH3A, CYP3A7, IDH3B CARM1 614/4885PRMT6 791/4885PRMT8 929/4885
US-20140350013-A1 INDAZOLES IDH3A, CYP3A7, IDH3B CARM1 614/4885PRMT6 791/4885PRMT8 929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.