SCHEMBL14720167

SCHEMBL14720167

CC(C)(C)[N+]1(C(=O)O)CC[C@@H](CNc2cccnc2)C1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
GRIN2B Q13224 1/20 0.46
CRHR1 P34998 1/20 0.42
GSK3A P49840 1/20 0.40
ALDH1A1 P00352 1/20 0.38
RAB9A P51151 4/20 0.37
NPC1 O15118 3/20 0.37
KDM4C Q9H3R0 2/20 0.37
NOTUM Q6P988 1/20 0.37
PKM P14618 1/20 0.36
VCP P55072 1/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
LMNA P02545 1/20 0.36
HIF1A Q16665 1/20 0.36
NAMPT P43490 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720215 0.81 GRIN2B (0.44) CYP3A4CYP2D6CYP2C9GRIN2BALDH1A1
SCHEMBL14720757 0.72 CHRM3 (0.44) CYP3A4CYP2D6CYP2C9TSHRLMNA
SCHEMBL13493771 0.69 CYP3A4 (0.49) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL14720234 0.68 GRIN2B (0.64) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL6778508 0.68 GBA1 (0.51) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL5870688 0.66 ACKR3 (0.54) CYP3A4CYP2D6CYP2C9GRIN2BALDH1A1
SCHEMBL18228060 0.66 CYP3A4 (0.53) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL12531359 0.66 KDM1A (0.50) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL4037864 0.66 KCNH3 (0.56) CYP3A4CYP2D6CYP2C9GRIN2BCRHR1
SCHEMBL12622711 0.64 CA12 (0.50) RAB9ANPC1NOTUMPKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013028445-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed