SCHEMBL14720191

SCHEMBL14720191

CC(c1ccc(Br)cc1F)N1CCC2(CC1)CN(C1CC1)C(=O)CO2

nearest known ligand 0.46

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 7/20 0.46
FASN P49327 4/20 0.40
HSD11B1 P28845 7/20 0.39
APLNR P35414 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720349 0.87 FASN (0.38) OPRM1FASNHSD11B1
SCHEMBL14720433 0.86 FASN (0.36) OPRM1FASNHSD11B1APLNR
SCHEMBL14720613 0.86 FASN (0.37) OPRM1FASNHSD11B1
SCHEMBL14720420 0.85 FASN (0.36) OPRM1FASNHSD11B1
SCHEMBL14722456 0.85 FASN (0.45) OPRM1FASNHSD11B1
SCHEMBL14720313 0.84 HSD11B1 (0.45) OPRM1FASNHSD11B1
SCHEMBL14720419 0.84 FASN (0.36) OPRM1FASNHSD11B1
SCHEMBL14720239 0.83 FASN (0.36) OPRM1FASNHSD11B1
SCHEMBL14720839 0.83 FASN (0.34) OPRM1FASNHSD11B1APLNR
SCHEMBL14729648 0.80 FASN (0.64) OPRM1FASNHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2744333-B1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2016-10-05 EP disclosed
US-9084794-B2 Fatty acid synthase inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2015-07-21 US disclosed
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline Intellectual Property (No2) Limite (GB) 2014-07-10 US disclosed
EP-2744333-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2014-06-25 EP disclosed
WO-2013028447-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS FASN, FADS2, FADS1 OPRM1 3162/4885FASN 1/4885HSD11B1 381/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.