SCHEMBL14720313

SCHEMBL14720313

CC(c1ccc(Br)cc1)N1CCC2(CC1)CN(C1CC1)C(=O)CO2

nearest known ligand 0.45

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 17/20 0.45
OPRM1 P35372 2/20 0.41
FASN P49327 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720261 0.86 HSD11B1 (0.39) HSD11B1FASN
SCHEMBL14720191 0.84 OPRM1 (0.46) HSD11B1OPRM1FASN
SCHEMBL14720141 0.84 HSD11B1 (0.41) HSD11B1FASN
SCHEMBL14720346 0.80 HSD11B1 (0.36) HSD11B1FASN
SCHEMBL14720226 0.78 FASN (0.70) HSD11B1FASN
SCHEMBL15544411 0.77 SIGMAR1 (0.52) OPRM1FASN
SCHEMBL4536313 0.76 FASN (0.63) FASN
SCHEMBL14720314 0.76 SIGMAR1 (0.56) OPRM1FASN
SCHEMBL15543324 0.76 FASN (0.40) HSD11B1OPRM1FASN
SCHEMBL14722456 0.74 FASN (0.45) HSD11B1OPRM1FASN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2744333-B1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE IP NO 2 LTD (GB) 2016-10-05 EP disclosed
US-9084794-B2 Fatty acid synthase inhibitors GLAXOSMITHKLINE INTELLECTUAL PROPERTY (NO. 2) LIMITED (GB) 2015-07-21 US disclosed
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS GlaxoSmithKline Intellectual Property (No2) Limite (GB) 2014-07-10 US disclosed
EP-2744333-A1 FATTY ACID SYNTHASE INHIBITORS Glaxosmithkline Intellectual Property (No. 2) Limited (GB) 2014-06-25 EP disclosed
WO-2013028447-A1 FATTY ACID SYNTHASE INHIBITORS GLAXOSMITHKLINE LLC (US) 2013-02-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140194415-A1 FATTY ACID SYNTHASE INHIBITORS FASN, FADS2, FADS1 HSD11B1 381/4885OPRM1 3162/4885FASN 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.