SCHEMBL14720535

SCHEMBL14720535

BrCc1ccc(C=C2CCNCC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.36
HTR2C P28335 1/20 0.34
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32
PRKACA P17612 1/20 0.32
PRKACG P22612 1/20 0.32
PRKACB P22694 1/20 0.32
SRD5A1 P18405 1/20 0.31
HPGD P15428 1/20 0.30
IGF1R P08069 1/20 0.30
PIM1 P11309 1/20 0.30
PIM2 Q9P1W9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720429 0.81 HPGD (0.47) HRH3HTR2CTSHRPRKACAPRKACG
SCHEMBL14720582 0.81 HRH3 (0.37) HRH3HTR2CPRKACAPRKACGPRKACB
SCHEMBL18991965 0.81 IGF1R (0.47) HRH3HTR2CALDH1A1HPGDIGF1R
Hydrochloric Acid SCHEMBL4887847 0.80 OGA (0.36) HRH3HTR2CPRKACAPRKACGPRKACB
SCHEMBL20587570 0.79 OGA (0.40) HRH3HTR2CALDH1A1TSHRSRD5A1
SCHEMBL14730978 0.79 MAOA (0.43) HRH3HTR2CPRKACAPRKACGPRKACB
SCHEMBL7039734 0.77 HDAC3 (0.43) HRH3HTR2CALDH1A1TSHR
Hydrochloric Acid SCHEMBL14721151 0.77 HTR2C (0.43) HRH3HTR2CPRKACAPRKACGPRKACB
SCHEMBL12076004 0.75 PRKACA (0.41) HRH3HTR2CPRKACAPRKACGPRKACB
SCHEMBL20015685 0.75 IKBKB (0.48) HRH3HTR2CALDH1A1PIM1PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed