SCHEMBL14720622

SCHEMBL14720622

C(=C1CCNCC1)c1ccc(COc2cccnn2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
HTR2C P28335 2/20 0.34
HTR2B P41595 1/20 0.34
HTR2A P28223 1/20 0.34
RXRA P19793 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
HTR1A P08908 2/20 0.32
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
PRKACA P17612 1/20 0.32
PRKACG P22612 1/20 0.32
PRKACB P22694 1/20 0.32
HPGD P15428 5/20 0.32
PTPN1 P18031 2/20 0.32
POLB P06746 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720972 0.78 HRH3 (0.42) HDAC1HDAC6HDAC5RXRAGRIN1
SCHEMBL13278903 0.74 PTPN1 (0.56) HDAC6SLC6A2SLC6A3HPGDPTPN1
SCHEMBL4273423 0.72 LTA4H (0.47) HDAC1HDAC6HDAC5SLC6A2SLC6A3
SCHEMBL14720429 0.68 HPGD (0.47) HTR2CHTR2BPRKACAPRKACGPRKACB
SCHEMBL18991965 0.68 IGF1R (0.47) HTR2CHPGD
SCHEMBL14720582 0.68 HRH3 (0.37) HTR2CPRKACAPRKACGPRKACB
SCHEMBL14720535 0.68 HRH3 (0.36) HTR2CPRKACAPRKACGPRKACBHPGD
Hydrochloric Acid SCHEMBL4887847 0.67 OGA (0.36) HTR2CHTR2BPRKACAPRKACGPRKACB
SCHEMBL20587570 0.65 OGA (0.40) HTR2CHPGD
SCHEMBL1382507 0.65 HTR2C (0.52) HTR2CHTR2BPRKACAPRKACGPRKACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed