SCHEMBL14722994

SCHEMBL14722994

Cc1nn(C)c(C)c1-c1ccc(C=C2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.42
BRD4 O60885 1/20 0.42
CREBBP Q92793 1/20 0.42
GPR119 Q8TDV5 14/20 0.41
PIK3CD O00329 1/20 0.39
PTPN2 P17706 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN6 P29350 1/20 0.37
SMPD3 Q9NY59 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18280165 0.79 USP30 (0.47) GRM5GPR119PTPN2PTPN1PTPN6
SCHEMBL4635083 0.76 GRM5 (0.46) GRM5GPR119
SCHEMBL1870570 0.76 NR1H2 (0.54) GRM5GPR119PTPN2PTPN1PTPN6
SCHEMBL5497099 0.76 MEN1 (0.55) GRM5
SCHEMBL14720896 0.76 GRM5 (0.46) GRM5GPR119
SCHEMBL1473227 0.76 GPR119 (0.51) GRM5GPR119
SCHEMBL15699606 0.75 ALDH1A1 (0.54) GRM5GPR119
SCHEMBL20304919 0.75 SRD5A2 (0.55) GRM5GPR119
SCHEMBL16113569 0.74 MAPT (0.54) GRM5GPR119
SCHEMBL31701014 0.74 PTPN2 (0.46) GRM5GPR119PTPN2PTPN1PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed