SCHEMBL14724467

SCHEMBL14724467

Nc1ccc(CC2(C(=O)NCc3ccccc3Cl)CCNCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
METAP2 P50579 1/20 0.46
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 2/20 0.41
AKT2 P31751 1/20 0.41
HSD17B2 P37059 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TP53 P04637 1/20 0.40
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170740 0.91 KMT2A (0.54) NPC1RAB9AMETAP2KMT2AMEN1
SCHEMBL2172656 0.78 ATM (0.57) METAP2KMT2AMEN1L3MBTL1
SCHEMBL2170887 0.77 ATM (0.52) METAP2KMT2AMEN1ALDH1A1TP53
SCHEMBL1346681 0.76 NPC1 (0.63) NPC1RAB9AMETAP2KMT2AMEN1
SCHEMBL4726588 0.75 RAB9A (0.46) NPC1RAB9AMETAP2KMT2AMEN1
SCHEMBL7917175 0.73 ATM (0.53) METAP2ALDH1A1HTT
SCHEMBL4794131 0.72 SMN1; SMN2 (0.41) NPC1RAB9APOLBALDH1A1L3MBTL1
SCHEMBL2173199 0.72 ATM (0.52) NPC1RAB9AMETAP2KMT2APOLB
SCHEMBL7924596 0.72 TACR1 (0.49)
SCHEMBL2467978 0.72 METAP2 (0.47) NPC1RAB9AMETAP2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346848-B1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS HOFFMANN LA ROCHE (CH) 2013-02-27 EP disclosed