SCHEMBL7924596

SCHEMBL7924596

O=C(NCc1ccc(Cl)c(C(F)(F)F)c1)C1(Cc2ccccc2)CCNCC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.49
P2RX7 Q99572 7/20 0.46
TRPV1 Q8NER1 1/20 0.43
GRIN2B Q13224 1/20 0.43
ATM Q13315 1/20 0.43
FAAH O00519 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41
SLC6A3 Q01959 1/20 0.41
PPARG P37231 1/20 0.40
PPARA Q07869 1/20 0.40
AURKA O14965 2/20 0.40
RPS6KB1 P23443 2/20 0.40
CHRM3 P20309 1/20 0.40
EPHX2 P34913 1/20 0.40
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2172656 0.82 ATM (0.57) TACR1ATMSLC6A2SLC6A4SLC6A3
SCHEMBL2170887 0.81 ATM (0.52) TACR1ATMSLC6A2SLC6A4SLC6A3
SCHEMBL2173199 0.79 ATM (0.52) TACR1ATMSLC6A2SLC6A4SLC6A3
SCHEMBL7917175 0.77 ATM (0.53) TACR1TRPV1ATMSLC6A2SLC6A4
SCHEMBL2170262 0.76 CYP17A1 (0.52) ATMNAMPT
Trifluoroacetic Acid SCHEMBL31716872 0.75 P2RX7 (0.46) TACR1P2RX7TRPV1FAAHCA1
SCHEMBL2170740 0.73 KMT2A (0.54) EPHX2
SCHEMBL7921565 0.73 ALDH1A1 (0.51) TACR1ATMSLC6A2SLC6A4SLC6A3
SCHEMBL15682792 0.73 P2RX7 (0.57) P2RX7TRPV1CA1CA2CA7
SCHEMBL14724467 0.72 NPC1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010054968-A1 QUINAZOLINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2010-05-20 WO disclosed