SCHEMBL14725252

SCHEMBL14725252

C=Cc1c(OC)c(OC)cc2c1OCC(=O)C=C2c1ccc(OC)c(OC(=O)C(CC(C)C)NC(=O)C(O)C(N)Cc2ccccc2)c1

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 3/20 0.38
IL1RN P18510 11/20 0.36
ERAP2 Q6P179 11/20 0.36
ERAP1 Q9NZ08 9/20 0.36
PSMB5 P28074 2/20 0.34
CTSD P07339 1/20 0.34
BIRC2 Q13490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721273 0.94 METAP2 (0.40) METAP2IL1RNERAP2ERAP1PSMB5
SCHEMBL14725404 0.88 PSMB5 (0.36) IL1RNERAP2ERAP1PSMB5BIRC2
SCHEMBL14725258 0.84 METAP2 (0.40) METAP2IL1RNERAP2ERAP1PSMB5
SCHEMBL14721499 0.83 PSEN1 (0.40)
Carbamic Acid SCHEMBL14722093 0.77 SRC (0.39)
SCHEMBL14721711 0.76 GSK3B (0.36)
SCHEMBL14725254 0.75 METAP2 (0.42) METAP2IL1RNERAP2ERAP1PSMB5
SCHEMBL14725272 0.75 METAP2 (0.41) METAP2IL1RNERAP2ERAP1PSMB5
SCHEMBL14725494 0.73 PSEN1 (0.42)
SCHEMBL14722096 0.72 SRC (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed