SCHEMBL14725265

SCHEMBL14725265

COc1ccc(C2=CC(=O)CCc3c2cc(OC)c(OC)c3OC)cc1OC(=O)C(N)CC(C)C

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 3/20 0.38
FLT3 P36888 2/20 0.38
KDR P35968 1/20 0.38
PDK1 Q15118 1/20 0.36
AAK1 Q2M2I8 5/20 0.35
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
SLC10A2 Q12908 1/20 0.34
CIT O14578 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725510 1.00 GSK3B (0.38) GSK3BFLT3KDRPDK1AAK1
SCHEMBL14721711 0.85 GSK3B (0.36) GSK3BFLT3KDRPDK1AAK1
SCHEMBL14725450 0.84 AAK1 (0.43) AAK1CIT
SCHEMBL14721685 0.84 AAK1 (0.43) AAK1CIT
SCHEMBL14725511 0.83 SRC (0.40) AAK1KDM4EALDH1A1
SCHEMBL14725538 0.77 KDM4E (0.39) KDM4EALDH1A1HPGD
SCHEMBL14722148 0.76 TUBB4A (0.48) KDM4EALDH1A1HPGD
SCHEMBL14721851 0.76 TUBB4A (0.48) FLT3KDRKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL14722766 0.75 TUBB4A (0.47) KDM4EALDH1A1HPGD
SCHEMBL14725545 0.74 AAK1 (0.35) GSK3BFLT3KDRAAK1CIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed