SCHEMBL14725511

SCHEMBL14725511

COc1ccc(C2=CC(=O)CCc3c2cc(OC)c(OC)c3OC)cc1OC(=O)[C@H](CC(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 1/20 0.40
ALDH1A1 P00352 4/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
MAPT P10636 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
GAA P10253 2/20 0.37
AAK1 Q2M2I8 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAP1LC3B Q9GZQ8 1/20 0.35
MAP1LC3A Q9H492 1/20 0.35
REN P00797 1/20 0.35
LMNA P02545 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GLA P06280 1/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
CTSL P07711 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725517 0.88 AAK1 (0.44) SRCALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL14725494 0.88 PSEN1 (0.42) REN
SCHEMBL14721276 0.87 SRC (0.41) SRCALDH1A1SMN1; SMN2MAPTNPC1
Carbamic Acid SCHEMBL14722093 0.85 SRC (0.39) SRCALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL14725510 0.83 GSK3B (0.38) ALDH1A1AAK1KDM4E
SCHEMBL14725265 0.83 GSK3B (0.38) ALDH1A1AAK1KDM4E
SCHEMBL14722096 0.81 SRC (0.37) SRCALDH1A1SMN1; SMN2MAPTNPC1
SCHEMBL14725529 0.78 MMP1 (0.35) ALDH1A1SMN1; SMN2MAPTGAAMEN1
SCHEMBL14725528 0.78 REN (0.40) REN
SCHEMBL14721499 0.77 PSEN1 (0.40) REN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed