SCHEMBL14730818

SCHEMBL14730818

Bc1ccc2[nH]c3c(c2c1)C(C)(C)CC3=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 2/20 0.44
KDM4E B2RXH2 9/20 0.43
ALDH1A1 P00352 7/20 0.43
LMNA P02545 6/20 0.36
HPGD P15428 4/20 0.36
HSD17B10 Q99714 2/20 0.36
MAPT P10636 4/20 0.32
MAPK1 P28482 3/20 0.32
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CCNB2 O95067 1/20 0.30
CDK1 P06493 1/20 0.30
CCNB1 P14635 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
CCNB3 Q8WWL7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16248397 0.82 LMNA (0.50) MAPKAPK2KDM4EALDH1A1LMNAHPGD
SCHEMBL14730815 0.80 MEN1 (0.44) MAPKAPK2KDM4EALDH1A1LMNAHPGD
SCHEMBL14731470 0.73 MAPKAPK2 (0.44) MAPKAPK2KDM4EALDH1A1LMNAHPGD
SCHEMBL14731471 0.70 MAPKAPK2 (0.33) MAPKAPK2
SCHEMBL14731462 0.69 LMNA (0.55) MAPKAPK2KDM4EALDH1A1LMNAHPGD
SCHEMBL3005560 0.66 KDM4E (0.46) MAPKAPK2KDM4EALDH1A1LMNAHPGD
SCHEMBL16248398 0.64 KIF11 (0.44) MAPKAPK2KDM4EALDH1A1HSD17B10MAPT
SCHEMBL14731469 0.64 MAPKAPK2 (0.31) MAPKAPK2
SCHEMBL14730689 0.64 KDM4E (0.47) MAPKAPK2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL14730760 0.64 KDM4E (0.50) MAPKAPK2KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026163-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-28 WO disclosed
WO-2013026162-A1 HEPATITIS C INHIBITOR COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-02-28 WO disclosed