SCHEMBL14732144

SCHEMBL14732144

c1ncc(-c2ccc(NCCN3CCOCC3)nc2)[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.51
FYN P06241 3/20 0.50
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
ATR Q13535 1/20 0.47
SYK P43405 2/20 0.45
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2D6 P10635 3/20 0.44
LMNA P02545 2/20 0.44
CYP2C19 P33261 2/20 0.44
HSD17B10 Q99714 2/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
TLR9 Q9NR96 2/20 0.43
TP53 P04637 1/20 0.43
ALOX15 P16050 1/20 0.43
HIF1A Q16665 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3243091 0.79 CYP1A2 (0.64) KDRFYNNPC1RAB9AATR
SCHEMBL1256254 0.78 KDR (0.57) KDRFYNNPC1RAB9AATR
Hydrochloric Acid SCHEMBL1257055 0.77 KDR (0.56) KDRFYNNPC1RAB9AATR
SCHEMBL3249454 0.75 KDR (0.57) KDRFYNNPC1RAB9AATR
SCHEMBL2961915 0.75 BACE1 (0.51) KDRFYNNPC1RAB9AATR
SCHEMBL3383793 0.75 ATR (0.51) KDRFYNNPC1RAB9AATR
SCHEMBL29036797 0.75 FYN (0.60) KDRFYNNPC1RAB9AATR
SCHEMBL1256123 0.75 TSHR (0.60) KDRFYNNPC1RAB9ACYP1A2
SCHEMBL7936724 0.75 CYP3A4 (0.52) KDRFYNNPC1RAB9ACYP1A2
SCHEMBL31240694 0.75 CDK9 (0.49) KDRFYNCYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8389554-B2 Imidazothiadiazole derivatives MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 2013-03-05 US claimed