SCHEMBL3243091

SCHEMBL3243091

c1cncc(-c2ccc(NCCN3CCOCC3)nc2)c1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.64
CYP3A4 P08684 3/20 0.64
CYP2D6 P10635 3/20 0.64
CLK4 Q9HAZ1 1/20 0.64
KDR P35968 1/20 0.58
LMNA P02545 2/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
FYN P06241 2/20 0.53
ATR Q13535 1/20 0.53
DYRK1A Q13627 2/20 0.51
GSK3B P49841 1/20 0.51
WNT1 P04628 1/20 0.51
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
CYP2C19 P33261 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13356455 0.88 ACHE (0.59) CYP1A2CYP3A4CYP2D6CLK4KDR
SCHEMBL1256254 0.82 KDR (0.57) CYP1A2CYP3A4CYP2D6CLK4KDR
SCHEMBL21064292 0.82 KDR (0.55) CYP1A2CYP3A4CYP2D6CLK4KDR
Hydrochloric Acid SCHEMBL1257055 0.81 KDR (0.56) CYP1A2CYP3A4CYP2D6CLK4KDR
SCHEMBL15394542 0.80 KDR (0.57) CYP1A2CYP3A4CYP2D6CLK4KDR
SCHEMBL3249454 0.80 KDR (0.57) CYP1A2CYP3A4CYP2D6KDRLMNA
SCHEMBL14732144 0.79 KDR (0.51) CYP1A2CYP3A4CYP2D6CLK4KDR
SCHEMBL12978212 0.77 SMN1; SMN2 (0.53) LMNAMEN1KMT2A
SCHEMBL1944938 0.77 FYN (0.59) KDRFYN
SCHEMBL1256249 0.77 KDR (0.54) KDRFYNATRNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010057833-A1 COMPOUNDS FOR TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY BIOMARIN IGA, LTD. (BS) 2010-05-27 WO claimed
WO-2010057833-A1 COMPOUNDS FOR TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY BIOMARIN IGA, LTD. (BS) 2010-05-27 WO disclosed