SCHEMBL14732172

SCHEMBL14732172

N[SH](=O)=O.OCc1cc(-c2ccccc2)n(-c2ccccc2)n1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CA9 Q16790 13/20 0.68
CA1 P00915 12/20 0.68
CA2 P00918 12/20 0.68
PTGS2 P35354 4/20 0.64
CNR1 P21554 1/20 0.53
CNR2 P34972 1/20 0.53
RPA1 P27694 1/20 0.52
FAAH O00519 1/20 0.49
NPC1 O15118 1/20 0.49
RAB9A P51151 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13239860 0.91 CA1 (0.70) CA9CA1CA2PTGS2CNR1
SCHEMBL6344401 0.81 CA9 (1.00) CA9CA1CA2PTGS2
SCHEMBL12285042 0.81 PTGS2 (0.70) CA9CA1CA2PTGS2CNR1
SCHEMBL13352312 0.81 CA1 (0.60) CA9CA1CA2PTGS2CNR1
Sulfamide SCHEMBL7182772 0.80 PTGS2 (0.76) CA9CA1CA2PTGS2
SCHEMBL8689665 0.79 CA9 (1.00) CA9CA1CA2PTGS2
SCHEMBL3864236 0.79 PTGS2 (0.90) CA9CA1CA2PTGS2
SCHEMBL9941289 0.79 PTGS2 (1.00) CA9CA1CA2PTGS2
SCHEMBL3865949 0.78 PTGS2 (0.58) CA9CA1CA2PTGS2CNR1
SCHEMBL27710506 0.77 CNR1 (0.53) CA9CA1CA2PTGS2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44048-E1 4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyrazol-1-YL]benzenesulfonamide for the treatment of inflammation or an inflammation-associated disorder G.D. SEARLE LLC (US) 2013-03-05 US disclosed